YM471 (free base) [183173-00-4]

MedChem Express

YM471 (free base) [183173-00-4]

9

183173-00-4

Research Use Only

C39H38F2N4O3

648.74

YM471 free base is a non-peptide antagonist of vasopressin V1A and V2 receptors with potent and persistent antagonistic activity. YM471 exhibits high affinity for rat V1A and V2 receptors with K values of 0.16 and 0.77 nM, respectively[1].

O=C(C1=CC=C(C=C1)NC(C2=C(C3=CC=CC=C3)C=CC=C2)=O)N4C5=CC=CC=C5/C(C(F)(CC4)F)=C/C(N6CCC(CC6)N(C)C)=O

12352200