Zaldaride maleate

MedChem Express

Zaldaride maleate [109826-27-9]

10

109826-27-9

Research Use Only

98.0

C30H32N4O6

544.60

Zaldaride maleate (CGS-9343B) is a potent, orally active and selective inhibitor of calmodulin . Zaldaride maleate inhibits CaM (calmodulin)-stimulated cAMP phosphodiesterase activity, with an IC 50 of 3.3 nM [1] [2] . Zaldaride maleate prevents estrogen-induced transcription activation by ER, reversibly blocks voltage-activated Na + , Ca 2+ and K + currents in PC12 cells and inhibits nAChR [3] .

O=C(O)/C=C\C(O)=O.CC1(C2=CC=CN2C3=CC=CC=C3CO1)CN4CCC(N5C6=C(C=CC=C6)NC5=O)CC4

2°C to 8°C

12352200