ZEN-3219 [1952264-34-4]

MedChem Express

ZEN-3219 [1952264-34-4]

10

1952264-34-4

Research Use Only

99.75

C19H18N2O3

322.36

ZEN-3219 is a BET inhibitor with IC50s of 0.48, 0.16 and 0.47 microM for BRD4(BD1), BRD4(BD2) and BRD4(BD1BD2), respectively. ZEN-3219 can be used to form PROTACs to induce degradation of BRD4[1].

O=C(C=CC(C1=C(C)ON=C1C)=C2)N2CC3=CC=C(C4OC4)C=C3

-20°C,2°C to 8°C

12352200