![ZLD1039 [1826865-46-6] ZLD1039 [1826865-46-6]](https://www.targetmol.com/group3/M00/36/25/CgoaEGayOdKEDnUOAAAAAJWBdHg087.png)
ZLD1039 [1826865-46-6]
T29231
CAS Number1826865-46-6
Product group Chemicals
Estimated Purity99.82%
Molecular Weight612.8
Overview
- SupplierTargetMol Chemicals
- Product NameZLD1039 [1826865-46-6]
- Delivery Days Customer9
- CAS Number1826865-46-6
- CertificationResearch Use Only
- Chemical NameZLD1039
- Estimated Purity99.82%
- Molecular FormulaC36H48N6O3
- Molecular Weight612.8
- Scientific DescriptionZLD1039 is a potent, orally bioavailable EZH2 (Enhancer of Zeste Homolog 2) inhibitor with high selectivity. It demonstrates strong, concentration-dependent inhibition of both wild-type and mutant (Y641F and A677G) PRC2 (Polycomb Repressive Complex 2) enzymatic activities, exhibiting IC50 values of 5.6, 15, and 4.0 nM, respectively. Additionally, ZLD1039 effectively suppresses breast tumor growth and metastasis.
- Shelf life instruction3 years
- SMILESCCN(C1CCOCC1)c1cc(cc(C(=O)NCc2c3CCCCc3c(C)[nH]c2=O)c1C)-c1ccc(nc1)N1CCN(C)CC1
- Storage Instruction-20°C
- UNSPSC12352200