(5Z,2E)-CU-3 [1815598-71-0]

TargetMol Chemicals

(5Z,2E)-CU-3 [1815598-71-0]

10

1815598-71-0

Chemical

Research Use Only

(5Z,2E)-CU-3

99.02%

C16H12N2O4S3

392.47

(5Z,2E)-CU-3 is a potent and highly selective inhibitor of the DGKalpha isozyme with an IC50 value of 0.6 microM, competing with ATP and exhibiting a Km value of 0.48 mM. It specifically targets the catalytic region of DGKalpha without affecting the regulatory region and has demonstrated antitumor and immunogenic effects by promoting cancer cell apoptosis and T cell activation.

3 years

O=C1N(NS(=O)(=O)c2ccccc2)C(=S)S\C1=C/C=C/c1ccco1

-20°C

12352200