Bio-Connect

APS-2-79

HY-100627
MedChem Express
CAS Number2002381-25-9
Product group Chemicals
Estimated Purity99.38
Molecular Weight387.43
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Overview

  • Supplier
    MedChem Express
  • Product Name
    APS-2-79 [2002381-25-9]
  • Delivery Days Customer
    10
  • CAS Number
    2002381-25-9
  • Estimated Purity
    99.38
  • Molecular Formula
    C23H21N3O3
  • Molecular Weight
    387.43
  • Scientific Description
    APS-2-79 is a KSR -dependent MEK antagonist. APS-2-79 inhibits ATP biotin binding to KSR2 within the KSR2-MEK1 complexe with an IC 50 of 120 nM. APS-2-79 makes the stabilization of the KSR inactive state antagonizes oncogenic Ras-MAPK signaling [1] .
  • SMILES
    CC1=CC(OC2=CC=CC=C2)=CC=C1NC3=NC=NC4=CC(OC)=C(OC)C=C43
  • Storage Instruction
    -20°C,2°C to 8°C
  • UNSPSC
    12352200