AZ3976 [1418747-15-5]
HY-117724
CAS Number1418747-15-5
Product group Chemicals
Estimated Purity98.03
Molecular Weight317.34
Overview
- SupplierMedChem Express
- Product NameAZ3976 [1418747-15-5]
- Delivery Days Customer10
- CAS Number1418747-15-5
- CertificationResearch Use Only
- Estimated Purity98.03
- Molecular FormulaC15H19N5O3
- Molecular Weight317.34
- Scientific DescriptionAZ3976 is a potent plasminogen activator inhibitor type 1 (PAI-1) inhibitor with an IC50 value of 26 microM in an enzymatic chromogenic assay. AZ3976 is active with an IC50 of 16 microM in a plasma clot lysis assay. AZ3976 does not bind to active PAI-1 but bound reversibly to latent PAI-1. AZ3976 inhibits PAI-1 by enhancing the latency transition of active PAI-1. AZ3976 displays profibrinolytic activities in a human plasma clot lysis assay[1].
- SMILESO=C1N=C(NC2CN(C2)C(OC(C)(C)C)=O)NC3=NC=CC=C13
- Storage Instruction-20°C,2°C to 8°C
- UNSPSC12352200
![AZ3976 [1418747-15-5]](https://www.targetmol.com/group3/M00/02/EC/CgoaEWY7PHCEZlguAAAAALSucuo185.png)