BL-1249
ORB1089708
CAS Number18200-13-0
Product group Chemicals
Molecular Weight291.3503826
Overview
- SupplierBiorbyt
- Product NameBL-1249 [18200-13-0]
- Delivery Days Customer10
- CAS Number18200-13-0
- CertificationResearch Use Only
- Molecular FormulaC17H17N5
- Molecular Weight291.3503826
- Scientific DescriptionBL-1249 is a nonsteroidal anti-inflammatory drug (NSAID) and a potassium channel activator. BL-1249 exhibits more selective for the bladder (EC50 of 1.26 microM) than vascular tissue (EC50 of 21.0 microM). BL-1249 extracellular application activates all TREK subfamily members but has no effect on other K2P subfamilies. BL-1249 potently activates K2P2.1 (TREK-1) and K2P10.1 (TREK-2) with EC50 values of 5.5 microM and 8.0 microM, respectively
- SMILESN1N=NC(C2=CC=CC=C2NC2=CC=CC3CCCCC2=3)=N1
- UNSPSC12352200
![BL-1249 [18200-13-0]](https://www.targetmol.com/group3/M00/35/FE/CgoaEWayM-2ELtg-AAAAAJj0OlE574.png)