BMS-986122

Selleck Chemicals

BMS-986122

9

Research Use Only

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BMS-986122 is a selective, potent positive allosteric modulator of the mu-opioid receptor (micro-OR), shows potentiation of orthosteric agonist-mediated beta-arrestin recruitment, adenylyl cyclase inhibition, and G protein activation, and potentiates DAMGO-mediated [35S]GTPgammaS binding in mouse brain membranes.

12352200