BTRX-335140
M21654
CAS Number2244614-14-8
Product group Chemicals
Molecular Weight453.55
Overview
- SupplierAbMole BioScience
- Product NameBTRX-335140
- Delivery Days Customer9
- CAS Number2244614-14-8
- Category SupplierChemical
- CertificationResearch Use Only
- Molecular FormulaC25H32FN5O2
- Molecular Weight453.55
- Scientific DescriptionBTRX-335140 is a selective and orally active kappa opioid receptor (KOR) antagonist, has antagonist activity for kappaOR, uOR and deltaOR with IC50 values of 0.8 nM, 110 nM, and 6500 nM, respectively. Navacaprant endows with favorable in vitro ADMET and in vivo pharmacokinetic profiles and medication-like duration of action in rats.
- UNSPSC12352200