CMPD101 [865608-11-3]

HY-103045
Overview
- SupplierMedChem Express
- Product NameCMPD101 [865608-11-3]
- Delivery Days Customer5
- CAS Number865608-11-3
- CertificationResearch Use Only
- Estimated Purity98.95
- Molecular FormulaC24H21F3N6O
- Molecular Weight466.46
- Scientific DescriptionCMPD101 is a potent, highly selective and membrane-permeable small-molecule inhibitor of GRK2/3 with IC50 of 18 nM and 5.4 nM, respectively. CMPD101 exhibits less selectively against GRK1, GRK5, ROCK-2 and PKCalpha with IC50s of 3.1 microM , 2.3 microM, 1.4 microM and 8.1 microM, respectively. CMPD101 can be used for the study of heart failure[1].
- SMILESO=C(C1=CC(NCC2=NN=C(C3=CC=NC=C3)N2C)=CC=C1)NCC4=CC=CC=C4C(F)(F)F
- Storage Instruction-20°C,2°C to 8°C
- UNSPSC12352200