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CMPD101 [865608-11-3]

Research Use Only
HY-103045
MedChem Express
CAS Number865608-11-3
Product group Chemicals
Estimated Purity98.95
Molecular Weight466.46
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Overview

  • Supplier
    MedChem Express
  • Product Name
    CMPD101 [865608-11-3]
  • Delivery Days Customer
    5
  • CAS Number
    865608-11-3
  • Certification
    Research Use Only
  • Estimated Purity
    98.95
  • Molecular Formula
    C24H21F3N6O
  • Molecular Weight
    466.46
  • Scientific Description
    CMPD101 is a potent, highly selective and membrane-permeable small-molecule inhibitor of GRK2/3 with IC50 of 18 nM and 5.4 nM, respectively. CMPD101 exhibits less selectively against GRK1, GRK5, ROCK-2 and PKCalpha with IC50s of 3.1 microM , 2.3 microM, 1.4 microM and 8.1 microM, respectively. CMPD101 can be used for the study of heart failure[1].
  • SMILES
    O=C(C1=CC(NCC2=NN=C(C3=CC=NC=C3)N2C)=CC=C1)NCC4=CC=CC=C4C(F)(F)F
  • Storage Instruction
    -20°C,2°C to 8°C
  • UNSPSC
    12352200