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CMPD101 [865608-11-3]

CMPD101 [865608-11-3]

Research Use Only
T14989
TargetMol Chemicals
CAS Number865608-11-3
DownloadMSDS
Product group Chemicals
Estimated Purity99.01%
Molecular Weight466.46
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Overview

  • Supplier
    TargetMol Chemicals
  • Product Name
    CMPD101 [865608-11-3]
  • Delivery Days Customer
    4
  • CAS Number
    865608-11-3
  • Category Supplier
    Chemical
  • Certification
    Research Use Only
  • Chemical Name
    CMPD101
  • Estimated Purity
    99.01%
  • Molecular Formula
    C24H21F3N6O
  • Molecular Weight
    466.46
  • Scientific Description
    CMPD101 is a membrane-permeable small-molecule inhibitor of GRK2/3 (IC50: 18 nM and 5.4 nM). Which can be used for the study of heart failure. CMPD101 exhibits less selectively against GRK1, GRK5, ROCK-2 and PKCalpha with IC50s of 3.1 microM , 2.3 microM, 1.4 microM and 8.1 microM, respectively.
  • Shelf life instruction
    3 years
  • SMILES
    Cn1c(CNc2cccc(c2)C(=O)NCc2ccccc2C(F)(F)F)nnc1-c1ccncc1
  • Storage Instruction
    -20°C
  • UNSPSC
    12352200

References

  • Inhibition of prostatic smooth muscle contraction by the inhibitor of G protein-coupled receptor kinase 2/3, CMPD101. Yu Q et al., 2018 Jul 15, Eur J Pharmacol
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