CYP3cide [1390637-82-7]
HY-18642
CAS Number1390637-82-7
Product group Chemicals
Estimated Purity99.92
Molecular Weight456.59
Overview
- SupplierMedChem Express
- Product NameCYP3cide [1390637-82-7]
- Delivery Days Customer10
- CAS Number1390637-82-7
- CertificationResearch Use Only
- Estimated Purity99.92
- Molecular FormulaC26H32N8
- Molecular Weight456.59
- Scientific DescriptionCYP3cide (PF-4981517) is a potent, selective and time-dependent inhibitor of cytochrome P4503A4 (CYP3A4). The IC50 values for Midazolam 1-hydroxylase activity are 0.03 microM, 17 microM, and 71 microM for CYP3A4, CYP3A5, and CYP3A7, respectively. CYP3cide can be used to distinguish the contributions of CYP3A4 versus CYP3A5 on agent metabolism[1].
- SMILESCC1=CC=C(C2=C(C3=NN(C)C4=NC=NC(N5C[C@@H](N6CCCCC6)CC5)=C43)C=NN2C)C=C1
- Storage Instruction-20°C
- UNSPSC12352200
![PF-4981517 [1390637-82-7] [1390637-82-7]](https://www.targetmol.com/group3/M00/35/46/CgoaEGayGn-EPWBPAAAAAEfEFsY801.png)