PF-4981517 [1390637-82-7]
T21548
CAS Number1390637-82-7
Product group Chemicals
Estimated Purity99.77%
Molecular Weight456.59
Overview
- SupplierTargetMol Chemicals
- Product NamePF-4981517 [1390637-82-7]
- Delivery Days Customer9
- CAS Number1390637-82-7
- Category SupplierChemical
- CertificationResearch Use Only
- Chemical NamePF-4981517
- Estimated Purity99.77%
- Molecular FormulaC26H32N8
- Molecular Weight456.59
- Scientific DescriptionPF-4981517 (CYP3cide) is a efficient, specific and time-dependent inhibitor of cytochrome P4503A4 (CYP3A4). The IC 50 values for CYP3A activity are 0.03 microM,17 microM, and 71 microM for CYP3A4, CYP3A5, and CYP3A7, respectively. PF-4981517 is able to be used to distinguish the contributions of CYP3A4 versus CYP3A5 on drug Metabolism.
- Shelf life instruction3 years
- SMILESCc1ccc(cc1)-c1c(cnn1C)-c1nn(C)c2ncnc(N3CC[C@@H](C3)N3CCCCC3)c12
- Storage Instruction-20°C
- UNSPSC12352200