Endoxifen (Z-isomer)
M27811
CAS Number112093-28-4
Product group Chemicals
Molecular Weight373.49
Overview
- SupplierAbMole BioScience
- Product NameEndoxifen (Z-isomer)
- Delivery Days Customer9
- CAS Number112093-28-4
- Category SupplierChemical
- CertificationResearch Use Only
- Molecular FormulaC25H27NO2
- Molecular Weight373.49
- Scientific DescriptionEndoxifen Z-isomer is the most important Tamoxifen metabolite responsible for eliciting the anti-estrogenic effects of this drug in breast cancer cells expressing estrogen receptor-alpha (ERalfa). Endoxifen inhibits hERG tail currents at 50 mV in a concentration-dependent manner with IC50 values of 1.6 uM.
- UNSPSC12352200