Gartisertib [1613191-99-3]

TargetMol Chemicals

Gartisertib [1613191-99-3]

72

1613191-99-3

Research Use Only

Gartisertib

C25H29F2N9O3

541.55

ATR inhibitor 2 is an orally active, ATP-competitive, and selective ATR inhibitor (Ki <150 pM) with antitumor activity. ATR inhibitor 2 potently inhibits ATR-driven phosphorylated checkpoint kinase-1 (Chk1) phosphorylation (IC50: 8 nM).

3 years

Nc1nn2cc(F)cnc2c1C(=O)Nc1cncc(F)c1N1CCC(CC1)C(=O)N1CCN(CC1)C1COC1

-20°C

12352200