GNF4877
M14889
CAS Number2041073-22-5
Product group Chemicals
Molecular Weight494.52
Overview
- SupplierAbMole BioScience
- Product NameGNF4877
- Delivery Days Customer9
- CAS Number2041073-22-5
- Category SupplierChemical
- Molecular FormulaC25H27FN6O4
- Molecular Weight494.52
- Scientific DescriptionGNF4877 is a potent DYRK1A and GSK3bèta inhibitor with IC50s of 6 nM and 16 nM, respectively, which leads to blockade of nuclear factor of activated T-cells (NFATc) nuclear export and increased bèta-cell proliferation (EC50 of 0.66 uM for mouse bèta (R7T1) cells).
- UNSPSC12352200