GSK778
HY-136570
CAS Number2451862-42-1
Product group Chemicals
Estimated Purity98.93
Molecular Weight511.61
Overview
- SupplierMedChem Express
- Product NameGSK778 [2451862-42-1]
- Delivery Days Customer10
- CAS Number2451862-42-1
- CertificationResearch Use Only
- Estimated Purity98.93
- Molecular FormulaC30H33N5O3
- Molecular Weight511.61
- Scientific DescriptionGSK778 (iBET-BD1) is a potent and selective BD1 bromodomain inhibitor of the BET proteins, with IC50s of 75 nM (BRD2 BD1), 41 nM (BRD3 BD1), 41 nM (BRD4 BD1), and 143 nM (BRDT BD1), respectively. GSK778 phenocopies the effects of pan-BET inhibitors in cancer models[1].
- SMILESCC1=NOC(C)=C1C2=C(OC[C@@H]3CNCC3)C=C4C5=C(N=C(COC)N5[C@H](C)C6=CC=CC=C6)C=NC4=C2
- Storage Instruction-20°C,2°C to 8°C
- UNSPSC12352200
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Product group Chemicals
CAS Number2451862-42-1
Estimated Purity98.42%
Molecular Weight511.61
- SizePrice
Product group Chemicals
GSK778ORB1685237
CAS Number2451862-42-1
Estimated Purity98%
Molecular Weight511.61
- SizePrice