KDM5A-IN-1 [1905481-36-8]

TargetMol Chemicals

KDM5A-IN-1 [1905481-36-8]

9

1905481-36-8

Chemical

Research Use Only

KDM5A-IN-1

99.80%

C15H22N4O2

290.36

KDM5A-IN-1 is an orally available, potent and selective inhibitor of the pan-histidine lysine demethylase 5 KDM5, inhibiting KDM5A, KDM5B, and KDM5C with IC50 values of 45 nM, 56 nM, and 55 nM, respectively.KDM5A-IN-1 inhibits PC9 H3K4Me3, and may be useful in cancer research.

3 years

CC(C)c1cc([nH]n1)C(=O)N1CC[C@H](C1)NC(=O)C1CC1

-20°C

51202000