LP-935509
HY-117626
CAS Number1454555-29-3
Product group Chemicals
Estimated Purity99.74
Molecular Weight396.44
Overview
- SupplierMedChem Express
- Product NameLP-935509 [1454555-29-3]
- Delivery Days Customer10
- CAS Number1454555-29-3
- CertificationResearch Use Only
- Estimated Purity99.74
- Molecular FormulaC20H24N6O3
- Molecular Weight396.44
- Scientific DescriptionLP-935509 is an orally active, potent, selective, ATP-competitive and brain-penetrant inhibitor of adaptor protein-2 associated kinase 1 (AAK1) with an IC50 of 3.3 nM and a Ki of 0.9 nM, respectively. LP-935509 is also a potent inhibitor of BIKE (IC50=14 nM) and a modest inhibitor of GAK (IC50=320 nM). LP-935509 shows antinociceptive activity. LP-935509 can be used for neuropathic pain and SARS-CoV-2 research[1].
- SMILESO=C(N1CCN(C2=NC3=C(C4=CC=CN=C4OC)C=NN3C=C2)CC1)OC(C)C
- Storage Instruction-20°C,2°C to 8°C
- UNSPSC12352200