LY2183240
HY-10865
Overview
- SupplierMedChem Express
- Product NameLY2183240 [874902-19-9]
- Delivery Days Customer10
- CAS Number874902-19-9
- CertificationResearch Use Only
- Estimated Purity98.01
- Molecular FormulaC17H17N5O
- Molecular Weight307.35
- Scientific DescriptionLY2183240 is a highly potent blocker of anandamide uptake (IC50= 270 pM; Ki=540 nM). LY2183240 is a potent, covalent inhibitor of the endocannabinoid-degrading enzyme fatty acid amide hydrolase (FAAH) with an IC50 of 12.4 nM. LY2183240 inactivates FAAH by carbamylation of the enzymes serine nucleophile. LY2183240 also inhibits several other brain serine hydrolases with IC50s of 5.3, 0.09, 8.2 nM for MAG lipase, bh6 and KIAA1363, respectively[1][2] [3].
- SMILESO=C(N(C)C)N1N=NN=C1CC(C=C2)=CC=C2C3=CC=CC=C3
- Storage Instruction-20°C,2°C to 8°C
- UNSPSC12352200
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Product group Chemicals
LY2183240 [874902-19-9]T15802
CAS Number874902-19-9
Estimated Purity98.17%
Molecular Weight307.35
- SizePrice
Product group Chemicals
LY2183240ORB340588
CAS Number874902-19-9
Estimated Purity>98%
Molecular Weight307.35
- SizePrice
