LY2183240

AbMole BioScience

LY2183240

9

874902-19-9

Research Use Only

307.35

LY2183240 is a highly potent blocker of anandamide uptake (IC50= 270 pM; Ki=540 nM). LY2183240 is a potent, covalent inhibitor of the endocannabinoid-degrading enzyme fatty acid amide hydrolase (FAAH) with an IC50 of 12.4 nM.

CN(C)C(=O)[N]1N=NN=C1CC2=CC=C(C=C2)C3=CC=CC=C3

12352200