Bio-Connect

PF-6274484

HY-101450
MedChem Express
CAS Number1035638-91-5
Product group Chemicals
Estimated Purity98.76
Molecular Weight372.78
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Overview

  • Supplier
    MedChem Express
  • Product Name
    PF-6274484 [1035638-91-5]
  • Delivery Days Customer
    10
  • CAS Number
    1035638-91-5
  • Certification
    Research Use Only
  • Estimated Purity
    98.76
  • Molecular Formula
    C18H14ClFN4O2
  • Molecular Weight
    372.78
  • Scientific Description
    PF-6274484 is a potent EGFR inhibitor with K i s of 0.14 nM and 0.18 nM for EGFR-L858R/T790M and WT EGFR, respectively. PF-6274484 inhibits EGFR-L858R/T790M autophosphorylation in H1975 tumor cells and EGFR WT in A549 tumor cells with IC 50 s of 6.6 and 5.8 nM, respectively [1] .
  • SMILES
    C=CC(NC1=CC2=C(NC3=CC(Cl)=C(F)C=C3)N=CN=C2C=C1OC)=O
  • Storage Instruction
    -20°C,2°C to 8°C
  • UNSPSC
    12352200