Pralsetinib (BLU-667)

Selleck Chemicals

Pralsetinib (BLU-667) [2097132-94-8]

9

Research Use Only

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Pralsetinib (BLU-667, CS 3009, Gavreto) is a highly potent and selective RET (c-RET) inhibitor with an IC50 of 0.4 nM for WT RET. It also demonstrates potent activity (IC50 0.4 nmol/L) against common oncogenic RET alterations, including RET (M918T).

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