Sigma-1 receptor antagonist 3

MedChem Express

Sigma-1 receptor antagonist 3 [1639220-17-9]

5

1639220-17-9

Research Use Only

99.47

C19H23ClFN3O

363.86

Sigma-1 receptor antagonist 3 (compound135) is a potent and selective Sigma-1 (sigma1) receptor antagonist with a K i of 1.14 nM. Sigma-1 receptor antagonist 3 inhibits Human Ether-a-go-go-Related Gene (hERG) with an IC 50 of 1.54 microM. Sigma-1 receptor antagonist 3 has the potential for the neuropathic pain [1] .

CC1=NC(C2=CC=C(F)C=C2)=NC(OCCCN3CCCCC3)=C1Cl

-20°C,2°C to 8°C

12352200