Sigma-1 receptor antagonist 3 [1639220-17-9]

TargetMol Chemicals

Sigma-1 receptor antagonist 3

4

1639220-17-9

Chemical

Research Use Only

Sigma-1 receptor antagonist 3

C19H23ClFN3O

363.86

Sigma-1 receptor antagonist 3 is a more potent and selective antagonist of Sigma-1 (sigma1) receptor (Ki = 1.14 nM) than sigma2 receptor(Ki = 1239 nM). Sigma-1 receptor antagonist 3 inhibits Human Ether-a-go-go-Related Gene (hERG, IC50 = 1.54 microM)

3 years

Cc1nc(nc(OCCCN2CCCCC2)c1Cl)-c1ccc(F)cc1

-20°C

51202000