Talabostat

Biorbyt

Talabostat

16

149682-77-9

Research Use Only

C9H19BN2O3

214.072

Talabostat (PT-100, Val-boroPro) is a potent, nonselective, orally available inhibitor of post-proline cleaving serine proteases with Ki of 0.18 nM for DPP4, also potently inhibits DPP8/9 (IC50=1.5/0.76 nM), FAP, DPP2 and some other DASH family enzymes.

CC(C)C(N)C(=O)N1C(B(O)O)CCC1

12352200