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A-3 hydrochloride

E2506
Selleck Chemicals
Estimated Purity...
Product group Chemicals
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Overview

  • Supplier
    Selleck Chemicals
  • Product Name
    A-3 hydrochloride [78957-85-4]
  • Delivery Days Customer
    9
  • Certification
    Research Use Only
  • Estimated Purity
    ...
  • Scientific Description
    A-3 hydrochloride, a potent, cell-permeable, reversible, ATP-competitive non-selective antagonist of various kinases, againsts cAMP-dependent protein kinase (PKA) (Ki=4.3 microM), casein kinase II (CK2) (Ki=5.1 microM) and myosin light chain kinase (MLCK) (Ki=7.4 microM), also inhibits Protein Kinase C (PKC) and casein kinase I (CK1) with Ki values of 47 microM and 80 microM, respectively.
  • UNSPSC
    12352200

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