GSK046 [2474876-09-8]
T8932
CAS Number2474876-09-8
Product group Chemicals
Estimated Purity99.97%
Molecular Weight414.47
Overview
- SupplierTargetMol Chemicals
- Product NameGSK046 [2474876-09-8]
- Delivery Days Customer9
- CAS Number2474876-09-8
- Category SupplierChemical
- CertificationResearch Use Only
- Chemical NameGSK046
- Estimated Purity99.97%
- Molecular FormulaC23H27FN2O4
- Molecular Weight414.47
- Scientific DescriptionGSK046 (iBET-BD2) is a potent, selective, and orally active BD2 bromodomain inhibitor of the BET proteins, with IC50 values of 264 nM [BRD2 BD2], 98 nM [BRD3 BD2], 49 nM [BRD4 BD2], and 214 nM [BRDT BD2], respectively. It exhibits immunomodulatory activity.
- Shelf life instruction3 years
- SMILESC[C@H](Oc1cc(cc(F)c1NC(C)=O)C(=O)N[C@H]1CC[C@H](O)CC1)c1ccccc1
- Storage Instruction-20°C
- UNSPSC12352200