GSK180736A [817194-38-0]

TargetMol Chemicals

GSK180736A [817194-38-0]

4

817194-38-0

Chemical

Research Use Only

GSK180736A

98.16%

C19H16FN5O2

365.36

GSK180736A is an effective and selective GRK2 inhibitor (IC50: 0.77 microM) and >100-fold selectivity over other GRKs. It is a weak inhibitor of PKA (IC50: 30 microM), but highly effective against ROCK1 (IC50: 100 nM).

3 years

CC1=C(C(NC(=O)N1)c1ccc(F)cc1)C(=O)Nc1ccc2[nH]ncc2c1

-20°C

12352200